EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
   3.4.14.10 | -999 |
- |
more |
Ki-value above 5 mM: Met-Met-OH, Asp-Tyr-OH, PhCH2-Val-Nvl-OH, PhCH2OCO-Val-Nvl-OH, CH3-Nl2-Nle-OCH3. Ki-value above 3.0 mM: CH3-Nle-Nle-NHCH3, PhCH2-Nle-Nle-NHCH3, PhCH2OCO-Val-Nle-O(CH2)3CH3. Ki-value above 0.5 mM: CH3CO-Val-Nvl-OH |
647156 |
| 3.4.14.10 | 0.000007 |
- |
butabindide |
- |
665981 |
| 3.4.14.10 | 0.000011 |
- |
butabindide |
wild type enzyme, using 0.2 mM of substrate L-Ala-L-Ala-L-Phe-p-nitroanilide, in 100 mM potassium phosphate buffer, pH 7.5, containing 2 mM dithiothreitol, and 15% glycerol, at 37°C |
696417 |
| 3.4.14.10 | 0.000015 |
- |
butabindide |
wild type enzyme, using 0.02 mM of substrate L-Ala-L-Ala-L-Phe-p-nitroanilide, in 100 mM potassium phosphate buffer, pH 7.5, containing 2 mM dithiothreitol, and 15% glycerol, at 37°C |
696417 |
| 3.4.14.10 | 0.00008 |
- |
aminobutyryl-Pro-n-butylamide |
- |
665981 |
| 3.4.14.10 | 0.0001 |
- |
butabindide |
pH 7.5, 37°C |
647155 |
| 3.4.14.10 | 0.00014 |
- |
(2S)-aminobutyryl-4-cis-benzyl-L-proline n-butylamide |
- |
665981 |
| 3.4.14.10 | 0.00021 |
- |
butabindide |
- |
666630 |
| 3.4.14.10 | 0.00032 |
- |
(2S)-aminobutyryl-(4S)-fluoro-L-proline n-butylamide |
- |
665981 |
| 3.4.14.10 | 0.001 |
- |
Ile-Pro-Ile-OH |
- |
647156 |
