EC Number |
KM Value [mM] |
KM Value Maximum [mM] |
Substrate |
Reference |
---|
3.4.21.97 | -999 |
- |
2-[5-Amino-2-(4-fluoro-phenyl)-6-oxo-6H-pyrimidin-1-yl]-N-(1-benzyl-2-oxo-2-thiazol-2-yl-ethyl)-acetamide |
- |
650227 |
3.4.21.97 | 0.0042 |
- |
4-[[4'-(dimethylamino)phenyl]azo]-benzoyl-Arg-Gly-Val-Val-Asn-Ala-Ser-Ser-Arg-Leu-Ala-5-[(2-'aminoethyl)-amino]naphthalenesulfonic acid |
pH 7.2, 30°C, mutant enzyme A143Q/R232H |
653320 |
3.4.21.97 | 0.0051 |
- |
4-[[4'-(dimethylamino)phenyl]azo]-benzoyl-Arg-Gly-Val-Val-Asn-Ala-Ser-Ser-Arg-Leu-Ala-5-[(2-'aminoethyl)-amino]naphthalenesulfonic acid |
pH 7.2, 30°C, mutant enzyme A143Q/D217N |
653320 |
3.4.21.97 | 0.0078 |
- |
4-[[4'-(dimethylamino)phenyl]azo]-benzoyl-Arg-Gly-Val-Val-Asn-Ala-Ser-Ser-Arg-Leu-Ala-5-[(2-'aminoethyl)-amino]naphthalenesulfonic acid |
pH 7.2, 30°C, mutant enzyme A143Q/D227N |
653320 |
3.4.21.97 | 0.009 |
- |
4-(4'-dimethylaminophenazo)benzoic acid-RGVVNAS-2-aminobutanoyl-RLN-5-[(2'-aminoethyl)-amino]-naphthalene-1-sulfonic acid |
- |
95610 |
3.4.21.97 | 0.0101 |
- |
4-(4'-dimethylaminophenylazo)benzoyl-Arg-Gly-Val-Val-Asn-Ala-Ser-Ser-Arg-Leu-Ala-5-((2'-aminoethyl)amino)-naphthalene-1-sulfonic acid |
pH 7.2, 30°C, wild-typelike mutant enzyme A143Q |
650071 |
3.4.21.97 | 0.0107 |
- |
4-[[4'-(dimethylamino)phenyl]azo]-benzoyl-Arg-Gly-Val-Val-Asn-Ala-Ser-Ser-Arg-Leu-Ala-5-[(2-'aminoethyl)-amino]naphthalenesulfonic acid |
pH 7.2, 30°C, mutant enzyme A143Q |
653320 |
3.4.21.97 | 0.0118 |
0.0196 |
acetyl-Cys-tert-butylglycine-tert-butylglycine-Asn(Me)2-Ala-7-amido-4-methylcoumarin |
24°C |
650245 |
3.4.21.97 | 0.012 |
- |
4-[[4'-(dimethylamino)phenyl]azo]-benzoyl-Arg-Gly-Val-Val-Asn-Ala-Ser-Ser-Arg-Leu-Ala-5-[(2-'aminoethyl)-amino]naphthalenesulfonic acid |
pH 7.2, 30°C, mutant enzyme A143Q/L229R |
653320 |
3.4.21.97 | 0.0136 |
- |
4-[[4'-(dimethylamino)phenyl]azo]-benzoyl-Arg-Gly-Val-Val-Asn-Ala-Ser-Ser-Arg-Leu-Ala-5-[(2-'aminoethyl)-amino]naphthalenesulfonic acid |
pH 7.2, 30°C, mutant enzyme A143Q/S225Y/L229R |
653320 |