EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor  |
Reference |
|---|
    5.3.3.5 | 0.000028 |
- |
(-)-emopamil |
IC50: 28 nM for the liver enzyme |
653279 |
| 5.3.3.5 | 0.000034 |
- |
(-)-emopamil |
IC50: 34 nM for the brain enzyme |
653279 |
| 5.3.3.5 | 0.0017 |
- |
(1'R,3a'R,7a'R,1''R)-5-(N-benzylpiperidin-4-yl)-aminomethyl-7a'-methyl-1'-(1,5-dimethylhexyl)-5-nitrospiro[1,3-dioxane-2,4'-octahydroindene] |
pH and temperature not specified in the publication |
726836 |
| 5.3.3.5 | 0.0047 |
- |
(1'R,3a'R,7a'R,1''R)-5-(N-benzylpiperidin-4-yl)-N-methylaminomethyl-7a'-methyl-1'-(1,5-dimethylhexyl)-5-nitrospiro[1,3-dioxane-2,4'-octahydroindene] |
pH and temperature not specified in the publication |
726836 |
| 5.3.3.5 | 0.0045 |
- |
1',2',3',4'-tetrahydro-5-(N-benzylpiperidin-4-yl)-aminomethyl-5-nitro-6'-(4-methylpentyloxy)-spiro[1,3-dioxane-2,1'-naphthaline] |
pH and temperature not specified in the publication |
726836 |
| 5.3.3.5 | 0.00025 |
- |
2-[4-[(1Z)-1,2-diphenylbut-1-en-1-yl]phenoxy]-N,N-dimethylethanamine |
noncompetitive, IC50: 0.00025 mM |
653232 |
| 5.3.3.5 | 0.0042 |
- |
3beta-[2-(diethylamino)ethoxy]androst-5-en-17-one |
IC50: 0.0042 mM |
649702 |
| 5.3.3.5 | 0.0001 |
- |
AY9944 |
- |
690830 |
| 5.3.3.5 | 0.0011 |
- |
CuCl2 |
IC50: 0.0011 mM, ifenprodil-labled enzyme |
653279 |
| 5.3.3.5 | 0.0023 |
- |
CuCl2 |
IC50: 0.0023 mM, ifenprodil-labeled enzyme |
653279 |
