EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference  |
|---|
    3.6.1.12 | 0.000044 |
- |
benzimidazole |
pH and temperature not specified in the publication, recombinant enzyme |
755792 |
| 3.6.1.12 | 0.0011 |
- |
2-methyl-4-(3-phenyl[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)quinoline |
pH and temperature not specified in the publication, recombinant enzyme |
755792 |
| 3.6.1.12 | 0.0033 |
- |
methyl 2-(4-methoxyphenyl)-3-methyl-4-oxo-3,4-dihydro[1]benzopyrano[3,4-b]pyrrole-1-carboxylate |
pH and temperature not specified in the publication, recombinant enzyme |
755792 |
| 3.6.1.12 | 0.0148 |
- |
2-[2-[2-(2-aminoethoxy)ethoxy]ethoxy]ethyl 2-(4-methoxyphenyl)-3-methyl-4-oxo-1,2,3,3a,4,9b-hexahydro[1]benzopyrano[3,4-b]pyrrole-1-carboxylate |
pH and temperature not specified in the publication, recombinant enzyme |
755792 |
| 3.6.1.12 | 0.00028 |
- |
3-(2-chlorophenyl)-5-methyl-6-[4-[(pyrrolidin-1-yl)methyl]phenyl][1,2]oxazolo[5,4-d]pyrimidin-4(5H)-one |
pH and temperature not specified in the publication |
756185 |
| 3.6.1.12 | 0.00058 |
- |
2-methyl-N-(4-oxo-6,7,8,9-tetrahydro-4H-pyrimido[2,1-b][1,3]benzothiazol-3-yl)benzamide |
pH and temperature not specified in the publication |
756185 |
| 3.6.1.12 | 0.00085 |
- |
5-methyl-3-(pyridin-3-yl)-6-[4-[(pyrrolidin-1-yl)methyl]phenyl][1,2]oxazolo[4,5-c]pyridin-4(5H)-one |
pH and temperature not specified in the publication |
756185 |
| 3.6.1.12 | 0.00089 |
- |
1-[[4-(5-methyl-4-oxo-3-phenyl-4,5-dihydro[1,2]oxazolo[4,5-c]pyridin-6-yl)phenyl]methyl]pyrrolidine-2,5-dione |
pH and temperature not specified in the publication |
756185 |
| 3.6.1.12 | 0.0009 |
- |
6-[4-[(dimethylamino)methyl]phenyl]-5-methyl-3-phenyl[1,2]oxazolo[4,5-c]pyridin-4(5H)-one |
pH and temperature not specified in the publication |
756185 |
| 3.6.1.12 | 0.0012 |
- |
5-methyl-6-[4-[(morpholin-4-yl)methyl]phenyl]-3-phenyl[1,2]oxazolo[4,5-c]pyridin-4(5H)-one |
pH and temperature not specified in the publication |
756185 |
