EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.6.1.12 | 0.000046 |
- |
(2-((5,6-dichloro-2-methyl-4-nitro-1H-benzo[d]imidazol-1-yl)-methyl)phenyl)boronic acid |
pH 8.0, 22°C |
757386 |
3.6.1.12 | 0.0011 |
- |
(2-chlorophenyl)[4-[3-(cyclopropylamino)-4-nitrophenyl]piperazin-1-yl]methanone |
pH and temperature not specified in the publication |
756187 |
3.6.1.12 | 0.000082 |
- |
(3-((5,6-dichloro-2-methyl-4-nitro-1H-benzo[d]imidazol-1-yl)-methyl)phenyl)boronic acid |
pH 8.0, 22°C |
757386 |
3.6.1.12 | 0.000206 |
- |
(4-((4-nitro-2-(trifluoromethyl)-1H-benzo[d]imidazol-1-yl)-methyl)phenyl)boronic acid |
pH 8.0, 22°C |
757386 |
3.6.1.12 | 0.000027 |
- |
(4-((5,6-dichloro-2-cyclopropyl-4-nitro-1H-benzo[d]imidazol-1-yl)methyl)phenyl)boronic acid |
pH 8.0, 22°C |
757386 |
3.6.1.12 | 0.000248 |
- |
(4-((5,6-dichloro-2-methyl-1H-benzo[d]imidazol-1-yl)methyl)-phenyl)boronic acid |
pH 8.0, 22°C |
757386 |
3.6.1.12 | 0.000046 |
- |
(4-((5,6-dichloro-2-methyl-4-nitro-1H-benzo[d]imidazol-1-yl)-methyl)phenyl)boronic acid |
pH 8.0, 22°C |
757386 |
3.6.1.12 | 0.000529 |
- |
(4-((5,6-difluoro-2-methyl-4-nitro-1H-benzo[d]imidazol-1-yl)-methyl)phenyl)boronic acid |
pH 8.0, 22°C |
757386 |
3.6.1.12 | 0.0034 |
- |
1,3-dimethyl-8-[4-(2-thienylcarbonyl)-1-piperazinyl]-3,7-dihydro-1H-purine-2,6-dione |
pH and temperature not specified in the publication |
756187 |
3.6.1.12 | 0.000075 |
- |
1-(4-(1H-pyrazol-1-yl)benzyl)-5,6-dichloro-2-methyl-4-nitro-1H-benzo[d]imidazole |
pH 8.0, 22°C |
757386 |