EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.7.7.43 | -999 |
- |
CDP |
1 mM, 37°C, pH 8.5, 15 min, 14% inhibition |
706038 |
2.7.7.43 | -999 |
- |
saturated sulfo-CDP |
1 mM, 37°C, pH 8.5, 15 min, 55% inhibition |
706038 |
2.7.7.43 | -999 |
- |
saturated sulfo-UDP |
1 mM, 37°C, pH 8.5, 15 min, 35% inhibition |
706038 |
2.7.7.43 | -999 |
- |
saturated sulfo-UDP ester |
1 mM, 37°C, pH 8.5, 15 min, 24% inhibition |
706038 |
2.7.7.43 | -999 |
- |
sulfo-CDP |
1 mM, 37°C, pH 8.5, 15 min, 47% inhibition |
706038 |
2.7.7.43 | -999 |
- |
sulfo-CTP |
1 mM, 37°C, pH 8.5, 15 min, 39% inhibition |
706038 |
2.7.7.43 | -999 |
- |
sulfo-UDP |
1 mM, 37°C, pH 8.5, 15 min, 6% inhibition |
706038 |
2.7.7.43 | -999 |
- |
sulfo-UTP |
1 mM, 37°C, pH 8.5, 15 min, 33% inhibition |
706038 |
2.7.7.43 | 0.13 |
- |
2-deoxy-2,3-dehydro-N-acetylneuraminic acid |
at pH 8.5 and 37°C |
760608 |
2.7.7.43 | 8.8 |
- |
Ca2+ |
at pH 8.5 and 37°C |
760608 |