EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.22.52 | 0.000000087 |
- |
methyl N-[[2'-([(2S)-1-[(2'-aminobiphenyl-2-yl)amino]-1-oxo-3-phenylpropan-2-yl]carbamoyl)biphenyl-2-yl]carbonyl]-L-phenylalanyl-L-valinate |
pH and temperature not specified in the publication |
708257 |
3.4.22.52 | 0.000006 |
- |
2-methyl-N-[(2S)-1-oxo-3-phenylpropan-2-yl]-7,8-dihydro-2H-[1,4]dioxino[2,3-g][1,2]benzothiazine-3-carboxamide 1,1-dioxide |
pH and temperature not specified in the publication |
708257 |
3.4.22.52 | 0.0000075 |
- |
calpain inhibitor VI |
pH and temperature not specified in the publication |
709624 |
3.4.22.52 | 0.000008 |
- |
calpain inhibitor III |
pH and temperature not specified in the publication |
709624 |
3.4.22.52 | 0.00002 |
- |
N'-((1S,2R)-1-benzyl-3-[(3,5-dimethoxybenzyl)amino]-2-hydroxypropyl)-N,N-dipropylbenzene-1,3-dicarboxamide |
IC50: 20 nM |
667939 |
3.4.22.52 | 0.000023 |
- |
N-[(2S)-1-[[(3S)-2-hydroxytetrahydrofuran-3-yl]amino]-1-oxopentan-2-yl]-10H-phenothiazine-2-carboxamide |
pH and temperature not specified in the publication |
708257 |
3.4.22.52 | 0.000025 |
- |
methyl (2Z)-[(3S)-3-sec-butyl-1-oxo-2,3-dihydroisoquinolin-4(1H)-ylidene]acetate |
- |
679230 |
3.4.22.52 | 0.000025 |
- |
methyl (S,S,Z)-(3-sec-butyl-1-oxo-2,3-dihydro-1H-isoquinolin-4-ylidene)acetate |
pH and temperature not specified in the publication |
709659 |
3.4.22.52 | 0.000028 |
- |
N-[(2S)-1-oxo-3-phenylpropan-2-yl]-7,8-dihydro-2H-[1,4]dioxino[2,3-g][1,2,4]benzothiadiazine-3-carboxamide 1,1-dioxide |
pH and temperature not specified in the publication |
708257 |
3.4.22.52 | 0.000029 |
- |
4-fluorophenyl (2-[(3-([(2-ethyl-1,1-dioxido-3,4,7,8-tetrahydro-2H-[1,4]dioxino[2,3-g][1,2]benzothiazin-3-yl)carbonyl]amino)-2-oxo-4-phenylbutanoyl)amino]ethyl)amidosulfite |
IC50: 29 nM |
667939 |