EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.22.52 | 0.00088 |
- |
(2S)-2-[[(4-fluorophenyl)sulfonyl]amino]-N-[(3S)-2-hydroxytetrahydrofuran-3-yl]-3-methylbutanamide |
pH and temperature not specified in the publication |
708257 |
3.4.22.52 | 0.0007 |
- |
(2S,5S)-5-benzyl-6-hydroxy-2-(2-methylpropyl)morpholin-3-one |
pH and temperature not specified in the publication |
708257 |
3.4.22.52 | 0.000038 |
- |
(3S)-2-hydroxytetrahydrofuran-3-yl N-[(10H-phenothiazin-2-yloxy)acetyl]-L-threonyl-L-leucinate |
pH and temperature not specified in the publication |
708257 |
3.4.22.52 | 0.000089 |
- |
(3S)-2-hydroxytetrahydrofuran-3-yl N-[(2S)-2-[[(10H-phenothiazin-2-yloxy)acetyl]amino]butanoyl]-L-leucinate |
pH and temperature not specified in the publication |
708257 |
3.4.22.52 | 0.001 |
- |
(3S)-3-[[N-(10H-phenothiazin-2-ylcarbonyl)-L-norvalyl]amino]tetrahydrofuran-2-yl acetate |
IC50 above 0.001 mM, pH and temperature not specified in the publication |
708257 |
3.4.22.52 | 0.013 |
- |
(6S,9S,16R)-6-(hydroxymethyl)-9-(2-methylpropyl)-16-phenyl-2,15-dioxa-7,10,13-triazabicyclo[16.2.2]docosa-1(20),18,21-triene-8,11,14-trione |
pH and temperature not specified in the publication |
707136 |
3.4.22.52 | 0.0004 |
- |
(6S,9S,16R)-9-(2-methylpropyl)-8,11,14-trioxo-16-phenyl-2,15-dioxa-7,10,13-triazabicyclo[16.2.2]docosa-1(20),18,21-triene-6-carbaldehyde |
pH and temperature not specified in the publication |
707136 |
3.4.22.52 | 0.029 |
- |
(7S,10S,13S,26S)-13,26-dibenzyl-7-methyl-10-(propan-2-yl)-5,7,8,10,11,13,14,25,26,28-decahydrotetrabenzo[k,m,t,v][1,4,7,10,15,18]hexaazacyclotetracosine-6,9,12,15,24,27-hexone |
pH and temperature not specified in the publication |
708257 |
3.4.22.52 | 0.00022 |
- |
(7S,10S,17R)-10-(2-methylpropyl)-9,12,15-trioxo-17-phenyl-2,16-dioxa-8,11,14-triazabicyclo[17.2.2]tricosa-1(21),19,22-triene-7-carbaldehyde |
pH and temperature not specified in the publication |
707136 |
3.4.22.52 | 0.00175 |
- |
(7S,10S,17R)-7-(hydroxymethyl)-10-(2-methylpropyl)-17-phenyl-2,16-dioxa-8,11,14-triazabicyclo[17.2.2]tricosa-1(21),19,22-triene-9,12,15-trione |
pH and temperature not specified in the publication |
707136 |