EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
6.3.4.18 | -999 |
- |
1-deoxy-1-(7,8-dimethyl-2,4-dioxo-3,4-dihydrobenzo[g]pteridin-10(2H)-yl)pentitol |
0.081 mM with fixed ATP and bicarbonate concentrations, 0.122 mM with fixed aminoimidazole ribonucleotide and bicarbonate concentrations |
702643 |
6.3.4.18 | -999 |
- |
2-(2,3-dioxo-2,3-dihydro-1H-indol-1-yl)-N,N-diethylacetamide |
0.029 mM with fixed ATP and bicarbonate concentrations, 0.04 mM with fixed aminoimidazole ribonucleotide and bicarbonate concentrations |
702643 |
6.3.4.18 | -999 |
- |
ethyl 4-(2-[[(4-chlorophenyl)sulfonyl]methyl]-1,3-thiazol-4-yl)-1,2-oxazole-3-carboxylate |
0.062 mM with fixed ATP and bicarbonate concentrations, 0.043 mM with fixed aminoimidazole ribonucleotide and bicarbonate concentrations |
702643 |
6.3.4.18 | 1.2 |
- |
ATP |
mutant enzyme R271K, in 50 mM HEPES, pH 7.8, at 37°C |
727030 |
6.3.4.18 | 3.3 |
- |
ATP |
wild type enzyme, in 50 mM HEPES, pH 7.8, at 37°C |
727030 |