EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.22.52 | 0.0059 |
- |
ritonavir |
- |
644006 |
3.4.22.52 | 0.01 |
- |
ethyl 4-(4-bromophenyl)-3-([N-[5-(1,2-dithiolan-3-yl)pentanoyl]-L-leucyl]amino)-2-oxobutanoate |
IC50 above 0.01 mM, pH and temperature not specified in the publication |
708257 |
3.4.22.52 | 0.0000005 |
- |
acetyl-DPMSSTYIEELGKREVTIPPKYREL-NH2 |
pH 7.5, 12°C |
678542 |
3.4.22.52 | 0.0000006 |
- |
acetyl-SSTYIEELGKREVTIPPKYRELLA-NH2 |
pH 7.5, 12°C |
678542 |
3.4.22.52 | 0.0000008 |
- |
acetyl-DPMSSTYIEELGKREVTIPPKYR-NH2 |
pH 7.5, 12°C |
678542 |
3.4.22.52 | 0.0000022 |
- |
acetyl-TYIEELGKREVTIPPKYRELLA-NH2 |
pH 7.5, 12°C |
678542 |
3.4.22.52 | 0.000026 |
- |
acetyl-SSTYIEELGKREVTIPPKYR-NH2 |
pH 7.5, 12°C |
678542 |
3.4.22.52 | 0.000093 |
- |
acetyl-TYIEELGKREVTIPPKYR-NH2 |
pH 7.5, 12°C |
678542 |
3.4.22.52 | 0.0069 |
- |
acetyl-DPMSSTYIEELGK-NH2 |
pH 7.5, 12°C |
678542 |
3.4.22.52 | 0.0117 |
- |
acetyl-SSTYIEELGK-NH-(CH2O)2-CH2C(O)-TIPPKYR-NH2 |
pH 7.5, 12°C |
678542 |