EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.5.1.20 | -999 |
- |
more |
dihydropteroylpolyglutamate inhibitors with different numbers of glutamyl residues |
392152 |
1.5.1.20 | -999 |
- |
more |
enzyme inhibition kinetics |
760654 |
1.5.1.20 | 0.000013 |
- |
dihydropteroylhexaglutamate |
- |
392155 |
1.5.1.20 | 0.0027 |
- |
S-adenosylmethionine |
pH 6.6, 46°C, enzyme mutant HsMTHFR1-656 |
761998 |
1.5.1.20 | 0.0065 |
- |
dihydrofolate |
- |
392152 |
1.5.1.20 | 0.014 |
- |
NADH |
recombinant wild-type enzyme, pH 7.2, 4°C, the mutant enzymes all show a Km below 0.0035 mM |
654771 |
1.5.1.20 | 0.021 |
- |
S-adenosylmethionine |
pH 6.6, 46°C, enzyme mutant HsMTHFR38-644 |
761998 |
1.5.1.20 | 0.04 |
0.051 |
(+)-5-methyl-5,6,7,8-tetrahydropteroylpentaglutamate |
- |
437717 |
1.5.1.20 | 0.061 |
- |
methylenetetrahydrofolate |
recombinant wild-type enzyme, pH 7.2, 4°C |
654771 |
1.5.1.20 | 0.16 |
- |
5,10-methylenetetrahydrofolate |
mutant F223L, pH 7.2, 25°C |
696353 |