EC Number |
KM Value [mM] |
KM Value Maximum [mM] |
Substrate |
Reference |
---|
3.4.24.B14 | 0.023 |
- |
3-methoxysuccinyl-Gly-Leu-Phe-Met-7-amido-4-methylcoumarin |
37°C, membrane-bound form of NEP2 |
690798 |
3.4.24.B14 | 0.027 |
- |
succinyl-Ala-Ala-Phe-7-amido-4-methylcoumarin |
37°C, membrane-bound form of NEP2 |
690798 |
3.4.24.B14 | 0.035 |
- |
3-methoxysuccinyl-Gly-Leu-Phe-Met-7-amido-4-methylcoumarin |
37°C, secreted soluble form of NEP2 |
690798 |
3.4.24.B14 | 0.04 |
- |
succinyl-Ala-Ala-Phe-4-methylcoumarin 7-amide |
37°C, pH 7.2, mutant enzyme L739G |
669280 |
3.4.24.B14 | 0.04 |
- |
succinyl-Ala-Ala-Val-7-amido-4-methylcoumarin |
37°C, membrane-bound form of NEP2 |
690798 |
3.4.24.B14 | 0.044 |
- |
succinyl-Ala-Ala-Phe-4-methylcoumarin 7-amide |
37°C, pH 7.2, mutant enzyme L739G/S133G |
669280 |
3.4.24.B14 | 0.045 |
- |
succinyl-Ala-Ala-Phe-4-methylcoumarin 7-amide |
37°C, pH 7.2, mutant enzyme R131M |
669280 |
3.4.24.B14 | 0.05 |
- |
succinyl-Ala-Ala-Phe-7-amido-4-methylcoumarin |
37°C, secreted soluble form of NEP2 |
690798 |
3.4.24.B14 | 0.062 |
- |
succinyl-Ala-Ala-Phe-4-methylcoumarin 7-amide |
37°C, pH 7.2. wild-type enzyme |
669280 |
3.4.24.B14 | 0.1 |
- |
succinyl-Ala-Ala-Val-7-amido-4-methylcoumarin |
37°C, secreted soluble form of NEP2 |
690798 |