Inhibitors | Comment | Organism | Structure |
---|---|---|---|
3-isobutyl-methylxanthine | inhibitor of all PDE isoforms except PDE8 | Bos taurus | |
Cilostamide | inhibitor of isoform PDE3 | Bos taurus | |
additional information | the major enzyme activity (isoform PDE8) is insensitive towards 3-isobutyl-methylxanthine | Bos taurus | |
papaverine | inhibitor of isoform PDE10 | Bos taurus | |
rolipram | inhibitor of isoform PDE4 | Bos taurus |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
3',5'-cAMP + H2O | Bos taurus | - |
5'-AMP | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Bos taurus | - |
- |
- |
Purification (Comment) | Organism |
---|---|
HiTrap-Q Sepharose column chromatography | Bos taurus |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
epididymal fluid | - |
Bos taurus | - |
epididymis | - |
Bos taurus | - |
seminal plasma | - |
Bos taurus | - |
seminal vesicle | - |
Bos taurus | - |
spermatozoon | - |
Bos taurus | - |
testis | - |
Bos taurus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
3',5'-cAMP + H2O | - |
Bos taurus | 5'-AMP | - |
? |
Subunits | Comment | Organism |
---|---|---|
? | x * 60000, isoform PDE10 appears on SDS-PAGE as bands of 75000 and 60000 Da in size | Bos taurus |
? | x * 75000, isoform PDE10 appears on SDS-PAGE as bands of 75000 and 60000 Da in size | Bos taurus |
Synonyms | Comment | Organism |
---|---|---|
cAMP-PDE | - |
Bos taurus |
cAMP-phosphodiesterase | - |
Bos taurus |
PDE10A | isoform | Bos taurus |
PDE3 | isoform | Bos taurus |
PDE4 | isoform | Bos taurus |
PDE8 | isoform | Bos taurus |