EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   5.6.1.3 | 0.00000023 |
- |
docetaxel |
mutant D130V, pH 6.8 |
689127 |
| 5.6.1.3 | 0.0000003 |
- |
docetaxel |
wild-type, pH 6.8 |
689127 |
| 5.6.1.3 | 0.00000045 |
- |
6-[4-(trifluoromethyl)phenyl]-3,4-dihydroquinolin-2(1H)-one |
mutant D130V, pH 6.8 |
689127 |
| 5.6.1.3 | 0.00000046 |
- |
SB-731489 |
wild-type, pH 6.8 |
689127 |
| 5.6.1.3 | 0.000002 |
- |
3-(dimethylamino)-N-(((2R,4aS,5R,10bS)-9-isopropyl-5-phenyl-3,4,4a,5,6,10b-hexahydro-2H-pyrano[3,2-c]quinolin-2-yl)methyl)propane-1-sulfonamide |
pH and temperature not specified in the publication |
711401 |
| 5.6.1.3 | 0.000002 |
- |
N-(((2R,4aS,5R,10bS)-9-chloro-7-fluoro-5-phenyl-3,4,4a,5,6,10b-hexahydro-2H-pyrano[3,2-c]quinolin-2-yl)methyl)-2-(dimethylamino)ethanesulfonamide |
pH and temperature not specified in the publication |
711401 |
| 5.6.1.3 | 0.000003 |
- |
1-((2R,4aS,5R,10bS)-9-bromo-7-fluoro-5-phenyl-3,4,4a,5,6,10b-hexahydro-2H-pyrano[3,2-c]quinolin-2-yl)-N-methylmethanamine |
pH and temperature not specified in the publication |
711401 |
| 5.6.1.3 | 0.000004 |
- |
1-((2R,4aS,5R,10bS)-9-(tert-butyl)-5-phenyl-3,4,4a,5,6,10b-hexahydro-2H-pyrano[3,2-c]quinolin-2-yl)-N-methylmethanamine |
pH and temperature not specified in the publication |
711401 |
| 5.6.1.3 | 0.000004 |
- |
2-(methylamino)-N-(((2R,4aS,5R,10bS)-5-phenyl-9-(trifluoromethyl)-3,4,4a,5,6,10b-hexahydro-2H-pyrano[3,2-c]quinolin-2-yl)methyl)ethanesulfonothioamide |
pH and temperature not specified in the publication |
711401 |
| 5.6.1.3 | 0.000004 |
- |
4-((2R,4aS,5R,10bS)-2-((methylamino)methyl)-9-(trifluoromethyl)-3,4,4a,5,6,10b-hexahydro-2H-pyrano[3,2-c]quinolin-5-yl)phenol |
pH and temperature not specified in the publication |
711401 |
