EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.5.3.1 | 0.00005 |
- |
fungizone |
pH 9.5, 37°C, activity in promastigote |
754290 |
3.5.3.1 | 0.00022 |
- |
2-(S)-amino-6-boronohexanoic acid |
pH 9.5, 25°C, supramolecular tandem assay method |
704175 |
3.5.3.1 | 0.00032 |
- |
6-borono-2-[2-(pyrrolidin-1-yl)ethyl]norleucine |
arginase I, at pH 7.4 and 37°C |
733483 |
3.5.3.1 | 0.00037 |
- |
6-borono-2-[2-(4-hydroxypiperidin-1-yl)ethyl]norleucine |
arginase I, at pH 7.4 and 37°C |
733483 |
3.5.3.1 | 0.00052 |
- |
6-borono-2-[2-(diethylamino)ethyl]norleucine |
arginase I, at pH 7.4 and 37°C |
733483 |
3.5.3.1 | 0.00062 |
- |
6-borono-2-[2-(pyrrolidin-1-yl)ethyl]norleucine |
arginase II, at pH 7.4 and 37°C |
733483 |
3.5.3.1 | 0.000934 |
- |
6-borono-2-[2-(diethylamino)ethyl]norleucine |
arginase II, at pH 7.4 and 37°C |
733483 |
3.5.3.1 | 0.00098 |
- |
6-borono-2-[2-(4-hydroxypiperidin-1-yl)ethyl]norleucine |
arginase II, at pH 7.4 and 37°C |
733483 |
3.5.3.1 | 0.0013 |
- |
2-(S)-amino-6-boronohexanoic acid |
pH 8.0, 21°C |
752398 |
3.5.3.1 | 0.00135 |
- |
2-(aminomethyl)-6-borononorleucine |
arginase II, at pH 7.4 and 37°C |
733483 |