EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.24.65 | 0.000007 |
- |
trans-4-[([[4-(4'-acetylbiphenyl-4-yl)-5-fluorothiophen-2-yl]carbonyl]amino)methyl]cyclohexanecarboxylic acid |
pH and temperature not specified in the publication |
717350 |
3.4.24.65 | 0.000013 |
- |
(3R)-3-[([5-fluoro-4-[4-(pyridin-4-yl)phenyl]thiophen-2-yl]carbonyl)amino]-3-phenylpropanoic acid |
pH and temperature not specified in the publication |
717350 |
3.4.24.65 | 0.000024 |
- |
(3R)-3-([[4-(4'-acetylbiphenyl-4-yl)-5-fluorothiophen-2-yl]carbonyl]amino)-3-phenylpropanoic acid |
pH and temperature not specified in the publication |
717350 |
3.4.24.65 | 0.000085 |
- |
N-[(1R)-3-amino-3-oxo-1-phenylpropyl]-5-fluoro-4-[4-(trifluoromethoxy)phenyl]thiophene-2-carboxamide |
pH and temperature not specified in the publication |
717350 |
3.4.24.65 | 0.00014 |
- |
trans-4-[[([5-fluoro-4-[4-(trifluoromethoxy)phenyl]thiophen-2-yl]carbonyl)amino]methyl]cyclohexanecarboxylic acid |
pH and temperature not specified in the publication |
717350 |
3.4.24.65 | 0.0002 |
- |
(3R)-3-[([5-fluoro-4-[4-(trifluoromethoxy)phenyl]thiophen-2-yl]carbonyl)amino]-3-phenylpropanoic acid |
pH and temperature not specified in the publication |
717350 |
3.4.24.65 | 0.0004 |
- |
trans-4-[[([4-[4-(trifluoromethoxy)phenyl]thiophen-2-yl]carbonyl)amino]methyl]cyclohexanecarboxylic acid |
pH and temperature not specified in the publication |
717350 |
3.4.24.65 | 0.0036 |
- |
trans-4-[[([3-[4-(trifluoromethoxy)phenyl]-1,2-thiazol-5-yl]carbonyl)amino]methyl]cyclohexanecarboxylic acid |
pH and temperature not specified in the publication |
717350 |
3.4.24.65 | 0.031 |
- |
trans-4-[[([5-[4-(trifluoromethoxy)phenyl]-1,2-thiazol-3-yl]carbonyl)amino]methyl]cyclohexanecarboxylic acid |
pH and temperature not specified in the publication |
717350 |
3.4.24.65 | 0.954 |
- |
(1S,5S,7R)-3-biphenyl-4-ylmethyl-2-oxo-3-aza-6,8-dioxa-bicyclo[3.2.1]octane-7-carboxylic acid |
pH 7.0, 25°C, recombinant enzyme |
683226 |