EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.24.56 | 0.000015 |
- |
methyl [(2S)-2-[4-([5-[4-([(2S)-2-[(3S)-3-amino-2-oxopiperidin-1-yl]-2-cyclohexylacetyl]amino)phenyl]pentyl]oxy)phenyl]-3-(quinolin-3-yl)butyl]carbamate |
37°C, pH 7.5 |
754114 |
3.4.24.56 | 0.000018 |
- |
methyl [(2S)-2-(5-[5-[4-([(2S)-2-[(3S)-3-amino-2-oxopiperidin-1-yl]-2-cyclohexylacetyl]amino)phenyl]pentyl]-2-fluorophenyl)-3-(quinolin-3-yl)propyl]carbamate |
37°C, pH 7.5 |
754114 |
3.4.24.56 | 0.000022 |
- |
EWRF-cyclo(DGdPPEDap)LYLVCG-NH2 |
pH 7.5, 23°C |
754399 |
3.4.24.56 | 0.000044 |
- |
EWRF-cyclo(DGGGdPPEDap)LYLVCG-NH2 |
pH 7.5, 23°C |
754399 |
3.4.24.56 | 0.0000444 |
- |
InsL3 |
pH not specified in the publication, temperature not specified in the publication |
707150 |
3.4.24.56 | 0.0000537 |
- |
relaxin-3 |
pH not specified in the publication, temperature not specified in the publication |
707150 |
3.4.24.56 | 0.00006 |
- |
Ac-EWRFCGdPPECLYLVCG-NH2(Cys5-Cys10 disulfide) |
pH 7.5, 23°C |
754399 |
3.4.24.56 | 0.000077 |
- |
Ac-EWRFCGGGdPPECLYLVCG-NH2(Cys5-Cys12-disulfide) |
pH 7.5, 23°C |
754399 |
3.4.24.56 | 0.000086 |
- |
EWRFdPPEALYLV-NH2 |
pH 7.5, 23°C |
754399 |
3.4.24.56 | 0.0001 |
- |
((((S)-2-(1H-imidazol-4-yl)-1-methylcarbamoylethylcarbamoyl)-methyl)-(3-phenyl-propyl)-amino)-acetic acid |
in HEPES 50 mM, NaCl 100 mM, pH 7.4, at 37°C |
733788 |