EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.24.35 | -999 |
- |
more |
- |
683579 |
3.4.24.35 | 0.0000002 |
- |
ilomastat |
pH 7.4, 37°C |
717299 |
3.4.24.35 | 0.0000005 |
- |
(R)-2-(N-((6-fluoropyridin-3-yl)methyl)-4-methoxyphenyl-sulfonamido)-N-hydroxy-3-methylbutanamide |
- |
695847 |
3.4.24.35 | 0.0000005 |
- |
ilomastat |
- |
683230 |
3.4.24.35 | 0.000006 |
- |
CGS 27023A |
- |
695847 |
3.4.24.35 | 0.0000062 |
- |
5-[3-(hydroxymethyl)piperidin-1-yl]-5-(4-phenoxyphenyl)pyrimidine-2,4,6(1H,3H,5H)-trione |
pH 7.5, 37°C |
717980 |
3.4.24.35 | 0.0000081 |
- |
5-[4-(2-hydroxyethyl)piperazin-1-yl]-5-(4-phenoxyphenyl)pyrimidine-2,4,6(1H,3H,5H)-trione |
pH 7.5, 37°C |
717980 |
3.4.24.35 | 0.000012 |
- |
5-[4-(2-hydroxyethyl)piperidin-1-yl]-5-(4-phenoxyphenyl)pyrimidine-2,4,6(1H,3H,5H)-trione |
pH 7.5, 37°C |
717980 |
3.4.24.35 | 0.000017 |
- |
(2E)-3-(N-hydroxycarbamoyl)-2-isopropionyl-L-tryptophan-N-methylamide |
- |
683230 |
3.4.24.35 | 0.000026 |
- |
5-(1,5-dihydroxypentan-3-yl)-5-(4-phenoxyphenyl)pyrimidine-2,4,6(1H,3H,5H)-trione |
pH 7.5, 37°C |
717980 |