EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.22.B14 | 0.00046 |
- |
5-methylamino-2-methyl-N-[(R)-1-(1-naphthyl)ethyl]benzamide |
in 50 mM HEPES, pH 7.5 |
709449 |
3.4.22.B14 | 0.00056 |
- |
5-amino-2-methyl-N-[(R)-1-(1-naphthyl)ethyl]benzamide |
in 50 mM HEPES, pH 7.5 |
709449 |
3.4.22.B14 | 0.00056 |
- |
5-amino-2-methyl-N-[1-methyl-1-(1-naphthyl)ethyl]benzamide |
in 50 mM HEPES, pH 7.5 |
709449 |
3.4.22.B14 | 0.0013 |
- |
N-methyl-5-methylamino-2-methyl-N'-[(R)-1-(1-naphthyl)ethyl]benzamide |
in 50 mM HEPES, pH 7.5 |
709449 |
3.4.22.B14 | 0.0014 |
- |
2-methoxymethyl-5-nitrobenzoic acid methyl ester |
in 50 mM HEPES, pH 7.5 |
709449 |
3.4.22.B14 | 0.0023 |
- |
2-methyl-N-[(R)-1-(1-naphthyl)ethyl]benzamide |
in 50 mM HEPES, pH 7.5 |
709449 |
3.4.22.B14 | 0.00264 |
- |
5-N-acetylamino-2-methyl-N-[(R)-1-(1-naphthyl)ethyl]benzamide |
in 50 mM HEPES, pH 7.5 |
709449 |
3.4.22.B14 | 0.0027 |
- |
5-iodo-2-methyl-N-[1-methyl-1-(1-naphthyl)ethyl]benzamide |
in 50 mM HEPES, pH 7.5 |
709449 |
3.4.22.B14 | 0.0048 |
- |
5-N-tert-butoxycarbonylmethylamino-2-methyl-N'-[(R)-1-(1-naphthyl)ethyl]benzamide |
in 50 mM HEPES, pH 7.5 |
709449 |
3.4.22.B14 | 0.0052 |
- |
5-amino-2-methoxymethyl-N-[1-methyl-1-(1-naphthyl)ethyl]benzamide |
in 50 mM HEPES, pH 7.5 |
709449 |