EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.21.79 | 0.00008 |
- |
IEPD-CHO |
pH 7.4, 30°C |
732601 |
3.4.21.79 | 0.025 |
- |
2-[(5E)-5-[4-(2-amino-2-oxoethoxy)-3-methoxybenzylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]-N-(3,4-dimethylphenyl)acetamide |
pH 7.4, 30°C |
732601 |
3.4.21.79 | 0.028 |
- |
hydroxy(6-[2-methoxy-4-[(E)-(3-[2-[(4-methylphenyl)amino]-2-oxoethyl]-2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]phenoxy]pyridin-3-yl)oxoammonium |
pH 7.4, 30°C |
732601 |
3.4.21.79 | 0.035 |
- |
5-[2-(4-chlorophenoxy)ethoxy]-1-cyclohexyl-1H-tetrazole |
pH 7.4, 30°C |
732601 |
3.4.21.79 | 0.044 |
- |
2-[(4E)-4-[3-methoxy-4-(prop-2-yn-1-yloxy)benzylidene]-2,5-dioxoimidazolidin-1-yl]-N-(4-methylphenyl)acetamide |
pH 7.4, 30°C |
732601 |
3.4.21.79 | 0.044 |
- |
3-(4-chlorophenyl)-2-([[5-(2,3-dihydro-1,4-benzodioxin-2-yl)-4-phenyl-4,5-dihydro-3H-1,2,4-triazol-3-yl]sulfanyl]methyl)quinazolin-4(3H)-one |
pH 7.4, 30°C |
732601 |
3.4.21.79 | 0.045 |
- |
(3R)-N-cyclopropyl-1-(3-[[(3-methoxyphenyl)sulfonyl]amino]benzoyl)piperidine-3-carboxamide |
pH 7.4, 30°C |
732601 |