EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.21.117 | 0.00007 |
- |
2-(2-fluoro-phenyl)-5,6,7,8-tertrahydro-benzol[4,5]thieno[2,3-d][1,3]oxazin-4-one |
- |
699037 |
3.4.21.117 | 0.00039 |
- |
1-(2-bromobenzene-1-sulfonyl)-5-methyl-3-(2-methyl-4,5-dihydro-1H-imidazol-4-yl)-1H-indole |
pH not specified in the publication, temperature not specified in the publication |
753015 |
3.4.21.117 | 0.0004 |
- |
1-(2-bromobenzene-1-sulfonyl)-5-methyl-3-(2-methyl-4,5-dihydro-1H-imidazol-4-yl)-1H-indole |
pH not specified in the publication, temperature not specified in the publication |
753015 |
3.4.21.117 | 0.0012 |
- |
1-(2-chlorobenzene-1-sulfonyl)-5-methyl-3-(2-methyl-4,5-dihydro-1H-imidazol-4-yl)-1H-indole |
pH not specified in the publication, temperature not specified in the publication |
753015 |
3.4.21.117 | 0.0015 |
- |
1-(2-chlorobenzene-1-sulfonyl)-5-methyl-3-(2-methyl-4,5-dihydro-1H-imidazol-4-yl)-1H-indole |
pH not specified in the publication, temperature not specified in the publication |
753015 |
3.4.21.117 | 0.026 |
- |
LEKTI domain 6 |
- |
683785 |
3.4.21.117 | 0.0335 |
- |
(4S)-4-benzyl-2-(3,4-dimethoxyphenyl)-3,4-dihydro-5Hpyrido[10,20:1,2]imidazo [4,5-d][1,3]diazepin-5-one |
pH 8..0, 37°C |
731754 |
3.4.21.117 | 0.0557 |
- |
(4S)-4-benzyl-2-(3,4,5-trimethoxyphenyl)-3,4-dihydro-5Hpyrido[10,20:1,2] imidazo[4,5-d][1,3]diazepin-5-one |
pH 8..0, 37°C |
731754 |
3.4.21.117 | 0.057 |
- |
(4S)-4-benzyl-2-(2-methylphenyl)-3,4-dihydro-5H-pyrido[1',2':1,2]imidazo[4,5-d][1,3]diazepin-5-one |
pH 8..0, 37°C |
731754 |
3.4.21.117 | 0.068 |
- |
(4S)-4-benzyl-2-(4-methylphenyl)-3,4-dihydro-5H-pyrido[1',2':1,2]imidazo[4,5-d][1,3]diazepin-5-one |
pH 8..0, 37°C |
731754 |