EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.21.105 | 0.0004 |
- |
7-amino-3-butoxy-4-chloro-1H-isochromen-1-one |
pH 7.3, 37°C |
732744 |
3.4.21.105 | 0.00075 |
- |
7-amino-4-chloro-3-[(5-phenylpentyl)oxy]-1H-isochromen-1-one |
pH 7.3, 37°C |
732744 |
3.4.21.105 | 0.001 |
- |
2-(benzyloxy)-5-methyl-4H-3,1-benzoxazin-4-one |
pH not specified in the publication, temperature not specified in the publication |
753003 |
3.4.21.105 | 0.001 |
- |
N-[2-(cyclopropylmethoxy)phenyl]-3,3,3-trifluoro-2-(trifluoromethyl)propanamide |
25 mM HEPES, pH 7.4, 5 mM EDTA, 5% (v/v) glycerol, 0.5% (w/v) DDM, 20% (v/v) DMSO, at 25°C |
717016 |
3.4.21.105 | 0.0011 |
- |
7-amino-4-chloro-3-(2-phenylethoxy)-1H-isochromen-1-one |
pH 7.3, 37°C |
732744 |
3.4.21.105 | 0.0012 |
- |
2-(benzyloxy)-5-methyl-4H-3,1-benzoxazin-4-one |
pH not specified in the publication, temperature not specified in the publication |
753003 |
3.4.21.105 | 0.0013 |
- |
tert-butyl 2-[[3,3,3-trifluoro-2-(trifluoromethyl)propanoyl]amino]benzoate |
25 mM HEPES, pH 7.4, 5 mM EDTA, 5% (v/v) glycerol, 0.5% (w/v) DDM, 20% (v/v) DMSO, at 25°C |
717016 |
3.4.21.105 | 0.0016 |
- |
2-(benzyloxy)-5-methyl-4H-3,1-benzoxazin-4-one |
pH not specified in the publication, temperature not specified in the publication |
753003 |
3.4.21.105 | 0.0018 |
- |
N-[2-(cyclopentyloxy)phenyl]-3,3,3-trifluoro-2-(trifluoromethyl)propanamide |
25 mM HEPES, pH 7.4, 5 mM EDTA, 5% (v/v) glycerol, 0.5% (w/v) DDM, 20% (v/v) DMSO, at 25°C |
717016 |
3.4.21.105 | 0.0023 |
- |
3,3,3-trifluoro-N-[2-(propan-2-yloxy)phenyl]-2-(trifluoromethyl)propanamide |
25 mM HEPES, pH 7.4, 5 mM EDTA, 5% (v/v) glycerol, 0.5% (w/v) DDM, 20% (v/v) DMSO, at 25°C |
717016 |