EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.16.2 | 0.0000002 |
- |
[(3S,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidin-3-yl](4-[(1Z)-1-[(3-chloro-4-fluorophenyl)amino]-3-iminoprop-1-en-1-yl]piperidin-1-yl)methanone |
pH not specified in the publication, temperature not specified in the publication |
731430 |
3.4.16.2 | 0.0000002 |
- |
[4-[1-(3-chloro-4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl][(1R,2R,4S)-2-(2,4-difluorophenyl)-4-(dimethylamino)-4-methylcyclopentyl]methanone |
pH not specified in the publication, temperature not specified in the publication |
731431 |
3.4.16.2 | 0.0000003 |
- |
[(3S,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidin-3-yl](4-[(1Z)-1-[(2,5-dichlorophenyl)amino]-3-iminobut-1-en-1-yl]piperidin-1-yl)methanone |
pH not specified in the publication, temperature not specified in the publication |
731430 |
3.4.16.2 | 0.0000003 |
- |
[(3S,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidin-3-yl](4-[(1Z)-1-[(3-chloro-4-fluorophenyl)amino]-3-iminoprop-1-en-1-yl]piperidin-1-yl)methanone |
pH not specified in the publication, temperature not specified in the publication |
731430 |
3.4.16.2 | 0.0000003 |
- |
[4-[1-(3-chloro-4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl][(1R,2R,4S)-2-(2,4-difluorophenyl)-4-(dimethylamino)-4-methylcyclopentyl]methanone |
pH not specified in the publication, temperature not specified in the publication |
731431 |
3.4.16.2 | 0.0000004 |
- |
[(3S,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidin-3-yl](4-[(1Z)-1-[(2,5-dichlorophenyl)amino]-3-iminobut-1-en-1-yl]piperidin-1-yl)methanone |
pH not specified in the publication, temperature not specified in the publication |
731430 |
3.4.16.2 | 0.0000007 |
- |
2-[4-[3-(4-fluorophenyl)-1-methyl-1H-pyrazol-5-yl]-1-(2-phenylethyl)piperidin-4-yl]pyridine |
pH not specified in the publication, temperature not specified in the publication |
731447 |
3.4.16.2 | 0.0000033 |
- |
2-[4-[3-(4-fluorophenyl)-1-methyl-1H-pyrazol-5-yl]-1-(2-phenylethyl)piperidin-4-yl]pyridine |
pH not specified in the publication, temperature not specified in the publication |
731447 |
3.4.16.2 | 0.00004 |
- |
corn trypsin inhibitor |
IC50: 40 nM |
652251 |
3.4.16.2 | 0.00005 |
- |
diisopropyl fluorophosphonate |
IC50: 50 nM |
650716 |