EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.14.1 | -999 |
- |
N-[(1S)-1-cyano-2,2-dimethylpropyl]-3-thiophen-2-yl-L-alaninamide |
value above 0.003 mM |
707677 |
3.4.14.1 | -999 |
- |
N-[(1S)-1-cyano-2-(4-fluorophenyl)ethyl]-L-prolinamide |
value above 0.01 mM |
707677 |
3.4.14.1 | 0.0000003 |
- |
N-[(1S)-1-cyano-2-(5-phenylthiophen-2-yl)ethyl]-3-thiophen-2-yl-L-alaninamide |
- |
707677 |
3.4.14.1 | 0.0000007 |
- |
N-[(1S)-2-(1,3-benzothiazol-2-yl)-1-cyanoethyl]-3-thiophen-2-yl-L-alaninamide |
- |
707677 |
3.4.14.1 | 0.0000009 |
- |
N-[(1S)-1-cyano-2-phenylethyl]-3-thiophen-2-yl-L-alaninamide |
- |
707677 |
3.4.14.1 | 0.000001 |
- |
N-[(1S)-1-cyano-2-(naphthalen-2-yl)ethyl]-3-thiophen-2-yl-L-alaninamide |
- |
707677 |
3.4.14.1 | 0.0000017 |
- |
(4R)-N-[(1S)-1-cyano-2-phenylethyl]-4-(methylsulfanyl)-4-phenyl-L-prolinamide |
- |
707677 |
3.4.14.1 | 0.0000038 |
- |
N-[(1S)-1-cyano-2,2-diphenylethyl]-3-thiophen-2-yl-L-alaninamide |
- |
707677 |
3.4.14.1 | 0.0000051 |
- |
N-[(1S)-1-cyano-2-cyclohexylethyl]-3-thiophen-2-yl-L-alaninamide |
- |
707677 |
3.4.14.1 | 0.0000058 |
- |
N-[(1S)-1-cyano-2-(1H-indol-3-yl)ethyl]-3-thiophen-2-yl-L-alaninamide |
- |
707677 |