EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   3.2.1.166 | -999 |
- |
more |
dissociation constants, overview |
731468 |
| 3.2.1.166 | -999 |
- |
more |
IC50 values of heparan sulfate-mimicking glycopolymers, overview |
753249 |
| 3.2.1.166 | 0.000003 |
- |
roneparstat |
pH and temperature not specified in the publication |
753404 |
| 3.2.1.166 | 0.000005 |
- |
SST0001 |
pH 5.0 37°C, recombinant enzyme |
754394 |
| 3.2.1.166 | 0.00001 |
- |
(((2,2'-(((carbonylbis(azanediyl))bis(3-fluoro-4,1-phenylene))bis-(benzo[d]oxazole-2,5-diyl))bis(acetyl))bis(azanediyl))bis-(methylene))diboronic acid |
pH 5.0 37°C, recombinant enzyme |
754394 |
| 3.2.1.166 | 0.00002 |
- |
heparin |
heparanase action toward antithrombin-binding oligosaccharides |
692967 |
| 3.2.1.166 | 0.000025 |
- |
heparanase inhibitor PI-88 |
pH 5.0, 37°C |
701675 |
| 3.2.1.166 | 0.00005 |
- |
laminarin sulfate |
- |
694956 |
| 3.2.1.166 | 0.00008 |
- |
2,2'-((2,2'-(((thiocarbonylbis(azanediyl))bis(3-fluoro-4,1-phenylene))bis(benzo[d]oxazole-2,5-diyl))bis(acetyl))bis-(azanediyl))diacetic acid |
pH 5.0 37°C, recombinant enzyme |
754394 |
| 3.2.1.166 | 0.00018 |
- |
2,2'-(((carbonylbis(azanediyl))bis(3-fluoro-4,1-phenylene))bis-(benzo[d]oxazole-2,5-diyl))diacetic acid |
pH 5.0 37°C, recombinant enzyme |
754394 |
