EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
    3.1.1.1 | 0.00000021 |
- |
chlorpyrifos |
- |
691075 |
| 3.1.1.1 | 0.00000029 |
- |
paraoxon |
- |
691075 |
| 3.1.1.1 | 0.0000008 |
- |
paraoxon |
mutant L362D, 37°C, pH 7.4 |
678538 |
| 3.1.1.1 | 0.000001 |
- |
paraoxon |
mutant L362A, 37°C, pH 7.4 |
678538 |
| 3.1.1.1 | 0.0000013 |
- |
paraoxon |
wild-type, 37°C, pH 7.4 |
678538 |
| 3.1.1.1 | 0.00000158 |
- |
4-[7-[(diethoxyphosphoryl)oxy]-5-hydroxy-4-oxo-4H-chromen-3-yl]phenyl diethyl phosphate |
in 0.1 M sodium phosphate buffer, pH 7.0, at 30°C |
729570 |
| 3.1.1.1 | 0.00000179 |
- |
diethyl 5-hydroxy-4-oxo-2-phenyl-4H-chromen-7-yl phosphate |
in 0.1 M sodium phosphate buffer, pH 7.0, at 30°C |
729570 |
| 3.1.1.1 | 0.0000019 |
- |
paraoxon |
in 25 mM Tris-HCl (pH 8.0), at 25°C |
716466 |
| 3.1.1.1 | 0.00000249 |
- |
4-[7-[(diethoxyphosphoryl)oxy]-5-hydroxy-4-oxo-4H-chromen-2-yl]phenyl diethyl phosphate |
in 0.1 M sodium phosphate buffer, pH 7.0, at 30°C |
729570 |
| 3.1.1.1 | 0.0000031 |
- |
paraoxon |
mutant L362R, 37°C, pH 7.4 |
678538 |
