EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
    2.7.9.1 | 0 |
42 |
indirubin-3'-monoxime |
pH 8.0, 30°C |
762228 |
| 2.7.9.1 | 0.00076 |
- |
bisindolylmaleimide |
pH 8.0, 30°C |
762228 |
| 2.7.9.1 | 0.0015 |
- |
2-(1-(3-dimethylaminopropyl)-5-methoxyindol-3-yl)-3-(1H-indol-3-yl)maleimide |
pH 8.0, 30°C |
762228 |
| 2.7.9.1 | 0.0112 |
- |
N-[4-(3-amino-1H-indazol-4-yl)phenyl]-N'-(2-fluoro-5-methylphenyl)urea |
pH 8.0, 30°C |
762228 |
| 2.7.9.1 | 0.0162 |
- |
2-(4-amino-1-isopropyl-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-1H-indol-5-ol |
pH 8.0, 30°C |
762228 |
| 2.7.9.1 | 0.04 |
- |
unguinol |
- |
671485 |
| 2.7.9.1 | 0.113 |
- |
6-bromoindirubin-3'-monoxime |
pH 8.0, 30°C |
762228 |
| 2.7.9.1 | 0.29 |
- |
ilimaquinone |
- |
671485 |
| 2.7.9.1 | 0.292 |
- |
ilimaquinone |
uncompetitive/mixed type versus pyruvate and versus ATP, 48% inhibition of C4 acid cycle evolution. IC50: 0.292 mM |
661918 |
| 2.7.9.1 | 0.74 |
- |
2-hydroxy-5-methoxy-3-[[(1R,2S,4aS,8aS)-1,2,4a-trimethyl-5-methylenedecahydro-1-naphthalenyl]methyl]-1,4-benzoquinone |
pH 8.0, 30°C |
762228 |
