EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.7.1.67 | 0.00000098 |
- |
N-(2-((6-chloro-3-(4-methoxy-3-(morpholinosulfonyl)phenyl)-2-methylimidazo[1,2-b]pyridazin-8-yl)amino)ethyl)acetamide |
pH and temperature not specified in the publication |
759597 |
2.7.1.67 | 0.0000015 |
- |
KDU691 |
pH and temperature not specified in the publication |
759607 |
2.7.1.67 | 0.0000015 |
- |
N-(4-chlorophenyl)-N-methyl-3-[4-(methylcarbamoyl)phenyl]imidazo[1,2-a]pyrazine-6-carboxamide |
pH and temperature not specified in the publication |
758572, 759607 |
2.7.1.67 | 0.0000024 |
- |
N-(2-((6-chloro-3-(3-(N,N-dimethylsulfamoyl)-4-methoxyphenyl)-2-methylimidazo[1,2-b]pyridazin-8-yl)amino)ethyl)acetamide |
pH and temperature not specified in the publication |
759597 |
2.7.1.67 | 0.0000034 |
- |
5-[4-(methylsulfonyl)phenyl]-6'-(trifluoromethyl)-3,3'-bipyridin-2-amine |
pH and temperature not specified in the publication |
758572, 759607 |
2.7.1.67 | 0.0000034 |
- |
MMV390048 |
pH and temperature not specified in the publication |
759607 |
2.7.1.67 | 0.0000035 |
- |
2-[[7-(3,4-dimethoxyphenyl)quinoxalin-2-yl]amino]-N-methylacetamide |
pH and temperature not specified in the publication |
758572, 759607 |
2.7.1.67 | 0.0000035 |
- |
BQR695 |
pH and temperature not specified in the publication |
759607 |
2.7.1.67 | 0.0000053 |
- |
5-(6-chloro-8-[[(2-ethylpyridin-4-yl)methyl]amino]-2-methylimidazo[1,2-b]pyridazin-3-yl)-N-(1-hydroxybutan-2-yl)-2-methoxybenzene-1-sulfonamide |
pH and temperature not specified in the publication |
759597 |
2.7.1.67 | 0.0000061 |
- |
5-(6-chloro-8-[[(2-ethylpyridin-4-yl)methyl]amino]-2-methylimidazo[1,2-b]pyridazin-3-yl)-N-(2-hydroxyethyl)-2-methoxybenzene-1-sulfonamide |
pH and temperature not specified in the publication |
759597 |