EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.3.3.9 | -999 |
- |
16-ethenyl-21-oxo-19,20-didehydro-18-oxayohimban-17-yl hexopyranoside |
IC50 of 0.029 mg/ml |
735447 |
2.3.3.9 | -999 |
- |
3-ethenyl-2-(5-methoxy-9H-b-carbolin-1-yl)-1-methylcyclopentanol |
IC50 of 0.017 mg/ml |
735447 |
2.3.3.9 | -999 |
- |
9-(hydroxymethyl)-8-methyl-8,9,10,11,11a,12-hexahydro-6H-6,10:11,12a-dimethanoindolo[3,2-b]quinolizin-13-yl acetate |
IC50 of 0.021 mg/ml |
735447 |
2.3.3.9 | -999 |
- |
methyl 13-amino-2,11-dimethoxy-3-[(3,4,5-trimethoxybenzoyl)oxy]-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroindeno[2',1':3,4]pyrido[1,2-b]isoquinoline-1-carboxylate |
IC50 of 0.017 mg/ml |
735447 |
2.3.3.9 | -999 |
- |
pyruvate |
1 mM pyruvate: 40% activity |
702873 |
2.3.3.9 | -999 |
- |
pyruvate |
IC50 of 0.0048 mg/ml |
735447 |
2.3.3.9 | 0.05 |
- |
(1S,2S,3R)-2-(5-methoxy-9H-b-carbolin-1-yl)-1-methyl-3-(prop-1-en-2-yl)cyclopentanol |
at pH 7.0 and 35°C |
737048 |