EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.3.1.286 | 0.0001 |
0.001 |
6-chloro-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide |
pH 8.0, 37°C |
728857 |
2.3.1.286 | 0.0003 |
0.0026 |
suramin |
pH 8.0, 37°C |
728857 |
2.3.1.286 | 0.0008 |
- |
2-[1-[3-(amidinothio)propyl]-1H-indol-3-yl]-3-(1-methylindol-3-yl)maleimide methanesulfonate |
pH 8.0, 37°C |
728857 |
2.3.1.286 | 0.00102 |
- |
[histone H3]-thioacetyl-L-lysine |
at pH 7.5 and 25°C |
749884 |
2.3.1.286 | 0.0011 |
0.02 |
suramin |
pH 8.0, 37°C |
728857 |
2.3.1.286 | 0.0012 |
0.1 |
nicotinamide |
pH 8.0, 37°C |
728857 |
2.3.1.286 | 0.00145 |
- |
3-((2-methoxynaphthalen-1-yl)methyl)-7-((pyridin-3-ylmethyl)amino)-5,6,7,8-tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidin-4(3H)-one |
pH 7.5, temperature not specified in the publication |
729603 |
2.3.1.286 | 0.0019 |
- |
7-((3-methoxybenzyl)amino)-3-((2-methoxynaphthalen-1-yl)-methyl)-5,6,7,8-tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidin-4(3H)-one |
pH 7.5, temperature not specified in the publication |
729603 |
2.3.1.286 | 0.0034 |
- |
5-[4-[(4-bromobenzyl)oxy]benzylidene]-2-thioxodihydropyrimidine-4,6(1H,5H)-dione |
pH 8.0, 37°C |
728857 |
2.3.1.286 | 0.0035 |
- |
2-[1-[3-(amidinothio)propyl]-1H-indol-3-yl]-3-(1-methylindol-3-yl)maleimide methanesulfonate |
pH 8.0, 37°C |
728857 |