EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.3.1.129 | 0.00005 |
- |
WMLDPIAGKWSR |
pH 8.0, 30°C |
758450 |
2.3.1.129 | 0.00006 |
- |
peptide 920 |
forward reaction, pH 7.0, 22°C, versus TAMRA peptide |
720069 |
2.3.1.129 | 0.00014 |
- |
HM-UNAG peptide |
forward reaction, pH 7.0, 22°C, versus TAMRA peptide, in absence of holo-ACP |
720069 |
2.3.1.129 | 0.00015 |
- |
TAMRA peptide |
forward reaction, pH 7.0, 22°C |
720069 |
2.3.1.129 | 0.0002 |
- |
UDP-3-O-(R-3-hydroxymyristoyl)-N-acetylglucosamine |
pH 7.0, 22°C |
720069 |
2.3.1.129 | 0.000238 |
- |
HM-UNAG peptide |
forward reaction, pH 7.0, 22°C, versus TAMRA peptide, in presence of holo-ACP |
720069 |
2.3.1.129 | 0.00051 |
- |
peptide 920 |
forward reaction, pH 7.0, 22°C, versus TAMRA peptide, in presence of holo-ACP |
720069 |
2.3.1.129 | 0.0006 |
- |
peptide 920 |
forward reaction, pH 7.0, 22°C, versus 0.001 mM UNAG peptide |
720069 |
2.3.1.129 | 0.00073 |
- |
peptide 920 |
forward reaction, pH 7.0, 22°C, versus TAMRA peptide, in absence of holo-ACP |
720069 |
2.3.1.129 | 0.000923 |
- |
peptide 920 |
forward reaction, pH 7.0, 22°C, versus 5 mM UNAG peptide |
720069 |