EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.1.1.148 | 0.00069 |
- |
N-methyl-2-[4-[3-(3-oxo-2,3-dihydro-4H-1,4-benzoxazin-4-yl)propanoyl]piperazin-1-yl]-N-phenylacetamide |
pH 7.5, temperature not specified in the publication |
756483 |
2.1.1.148 | 0.00088 |
- |
N-[1-[3-(3-oxo-2,3-dihydro-4H-1,4-benzoxazin-4-yl)propanoyl]piperidin-4-yl]-N'-phenylurea |
pH 7.5, temperature not specified in the publication |
756483 |
2.1.1.148 | 0.00172 |
- |
4-(3-(3-oxo-2,3-dihydro-4H-pyrido[3,2-b][1,4]oxazin-4-yl)propanoyl)-N-phenylpiperazine-1-carboxamide |
pH 7.5, temperature not specified in the publication |
756483 |
2.1.1.148 | 0.0083 |
- |
5-undecyloxymethyl-2'-deoxyuridine 5'-monophosphate |
pH not specified in the publication, temperature not specified in the publication |
733512 |
2.1.1.148 | 0.00832 |
- |
5-undecyloxymethyl-2'-deoxyuridine 5'-monophosphate |
pH 7.5, 23° |
756170 |
2.1.1.148 | 0.016 |
- |
5,10-methylenetetrahydrofolate |
wild-type |
680675 |
2.1.1.148 | 0.048 |
- |
5,10-methylenetetrahydrofolate |
R182A mutant |
680675 |
2.1.1.148 | 93 |
- |
4-[3-(3-oxo-2,3-dihydro-4H-1,4-benzoxazin-4-yl)propanoyl]-N-phenylpiperazine-1-carboxamide |
pH 7.5, temperature not specified in the publication |
756483 |