EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.1.1.44 | 0.00072 |
- |
(-)-epigallocatechin gallate |
in 0.1 M Tris buffer (pH 7.5), 150 mM NaCl, 6 mM MgCl2, at 30°C |
685541 |
1.1.1.44 | 0.00121 |
- |
(-)-epicatechin gallate |
in 0.1 M Tris buffer (pH 7.5), 150 mM NaCl, 6 mM MgCl2, at 30°C |
685541 |
1.1.1.44 | 0.00128 |
- |
(-)-catechin gallate |
in 0.1 M Tris buffer (pH 7.5), 150 mM NaCl, 6 mM MgCl2, at 30°C |
685541 |
1.1.1.44 | 0.0013 |
- |
(5Z)-5-[[4-(3-fluorophenoxy)phenyl]methylidene]-2-imino-3-(2-methoxyphenyl)-1,3-thiazolidin-4-one |
25°C, pH 8.0 |
761698 |
1.1.1.44 | 0.0013 |
- |
MMV007199 |
pH 8.0, 25°C |
761698 |
1.1.1.44 | 0.00145 |
- |
(-)-gallocatechin gallate |
in 0.1 M Tris buffer (pH 7.5), 150 mM NaCl, 6 mM MgCl2, at 30°C |
685541 |
1.1.1.44 | 0.0016 |
- |
4,4'-[1,4-phenylenebis(oxy-1H-benzimidazole-6,2-diyl)]dianiline |
25°C, pH 8.0 |
761698 |
1.1.1.44 | 0.0016 |
- |
MMV011895 |
pH 8.0, 25°C |
761698 |
1.1.1.44 | 0.0018 |
- |
2,6-dimethoxy-4-[5-phenyl-4-[4-(phenylsulfanyl)phenyl]-1H-imidazol-2-yl]phenol |
25°C, pH 8.0 |
761698 |
1.1.1.44 | 0.0018 |
- |
5,6-bis(2H-1,3-benzodioxol-5-yl)-2-(3-methylphenyl)-4,7-diphenyl-3a,4,7,7a-tetrahydro-1H-4,7-methanoisoindole-1,3,8(2H)-trione |
25°C, pH 8.0 |
761698 |