EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.1.1.357 | 0.000037 |
- |
(5-methyl-1H-indol-2-yl)(4-propylpiperidin-1-yl)methanone |
pH 6.0, 22°C |
739797 |
1.1.1.357 | 0.00006 |
- |
Ursodeoxycholic acid |
recombinant enzyme, at pH 7.4 and 25°C |
724207 |
1.1.1.357 | 0.00007 |
- |
lithocholic acid |
native enzyme, at pH 7.4 and 25°C |
724207 |
1.1.1.357 | 0.00008 |
- |
lithocholic acid |
recombinant enzyme, at pH 7.4 and 25°C |
724207 |
1.1.1.357 | 0.00008 |
- |
Ursodeoxycholic acid |
native enzyme, at pH 7.4 and 25°C |
724207 |
1.1.1.357 | 0.00013 |
- |
chenodeoxycholic acid |
native enzyme, at pH 7.4 and 25°C |
724207 |
1.1.1.357 | 0.00015 |
- |
chenodeoxycholic acid |
recombinant enzyme, at pH 7.4 and 25°C |
724207 |
1.1.1.357 | 0.00029 |
- |
5-(benzenesulfonyl)-2-nitrophenol |
pH 6.0, 22°C |
739797 |
1.1.1.357 | 0.00049 |
- |
4-nitro-2-([4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]methyl)phenol |
pH 6.0, 22°C |
739797 |
1.1.1.357 | 0.0007 |
- |
Flufenamic acid |
recombinant enzyme, at pH 7.4 and 25°C |
724207 |