EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
4.1.3.36 | 0.4 |
- |
3-(2,4-dichlorophenyl)-3-oxopropyl-CoA |
above, pH 7.4, 25°C |
726554 |
4.1.3.36 | 0.027 |
- |
methyl (2Z)-(6-fluoro-2-oxo-2H-1,4-benzoxazin-3(4H)-ylidene)ethanoate |
non-competitive inhibitor Ki' = 0.0101 mM, pH not specified in the publication, temperature not specified in the publication |
714417 |
4.1.3.36 | 0.0463 |
- |
methyl (2Z)-(6-chloro-2-oxo-2H-1,4-benzoxazin-3(4H)-ylidene)ethanoate |
non-competitive inhibitor Ki' = 0.0185 mM, pH not specified in the publication, temperature not specified in the publication |
714417 |
4.1.3.36 | 0.01 |
- |
methyl (2Z)-(2-oxo-2H-1,4-benzoxazin-3(4H)-ylidene)ethanoate |
non-competitive inhibitor Ki' = 0.067 mM, pH not specified in the publication, temperature not specified in the publication |
714417 |
4.1.3.36 | 0.000103 |
- |
2-CoA-4-(2-chlorophenyl)-4-oxobutanoic acid |
pH 7.4, 25°C |
726554 |
4.1.3.36 | 0.000106 |
- |
2-CoA-4-(2,4-dichlorophenyl)-4-oxobutanoic acid |
pH 7.4, 25°C |
726554 |
4.1.3.36 | 0.000135 |
- |
2-CoA-4-(2-bromophenyl)-4-oxobutanoic acid |
pH 7.4, 25°C |
726554 |
4.1.3.36 | 0.000154 |
- |
2-CoA-4-(2-nitrophenyl)-4-oxobutanoic acid |
pH 7.4, 25°C |
726554 |
4.1.3.36 | 0.000204 |
- |
2-CoA-4-(2-fluorophenyl)-4-oxobutanoic acid |
pH 7.4, 25°C |
726554 |
4.1.3.36 | 0.000421 |
- |
2-CoA-4-(2-iodophenyl)-4-oxobutanoic acid |
pH 7.4, 25°C |
726554 |