EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.14.99.1 | 0.003 |
- |
alpha-linolenic acid |
inhibition of PGHS-2 |
676390 |
1.14.99.1 | 0.1226 |
- |
oleic acid |
inhibition of PGHS-2 |
676390 |
1.14.99.1 | 0.018 |
- |
quercetin |
isozyme PGHS-1, in 100 mM Tris-HCl buffer (pH 7.4), at 24°C |
701036 |
1.14.99.1 | 0.086 |
- |
quercetin |
isozyme PGHS-2, in 100 mM Tris-HCl buffer (pH 7.4), at 24°C |
701036 |
1.14.99.1 | 0.0388 |
- |
peroxynitrite |
peroxidase activity, enzyme is incubated with peroxynitrite in the presence of peroxides and arachidonic acid |
673809 |
1.14.99.1 | 0.0222 |
- |
peroxynitrite |
peroxidase activity, peroxynitrite is incubated with the resting enzyme and 30 s later, activity and protein nitration is analyzed |
673809 |
1.14.99.1 | 0.000041 |
- |
indomethacin |
pH 7.4, temperature not specified in the publication |
764274 |
1.14.99.1 | 0.0001 |
- |
N-butyl-5-[[(2,5-dihydroxyphenyl)methyl]amino]-2-hydroxybenzamide |
pH 7.4, temperature not specified in the publication |
764274 |
1.14.99.1 | 0.0001 |
- |
N-hexyl-5-[[(2,5-dihydroxyphenyl)methyl]amino]-2-hydroxybenzamide |
pH 7.4, temperature not specified in the publication |
764274 |
1.14.99.1 | 0.00011 |
- |
N-cyclohexyl-5-[(E)-[(2,5-dihydroxyphenyl)methylidene]amino]-2-hydroxybenzamide |
pH 7.4, temperature not specified in the publication |
764274 |