EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
6.3.3.6 | 0.005 |
- |
diphosphate |
pH 7.8, 22°C, variable substrate: (2S,5R)-carboxymethylproline, Ki(slope) |
721590 |
6.3.3.6 | 0.012 |
- |
diphosphate |
pH 7.8, 22°C, variable substrate: ATP, Ki(slope) |
721590 |
6.3.3.6 | 0.019 |
- |
diphosphate |
pH 7.8, 22°C, variable substrate: (2S,5R)-carboxymethylproline, Ki(intercept) |
721590 |
6.3.3.6 | 0.17 |
- |
AMP |
pH 7.8, 22°C, variable substrate: ATP, Ki(intercept) |
721590 |
6.3.3.6 | 0.28 |
- |
AMP |
pH 7.8, 22°C, variable substrate: (2S,5R)-carboxymethylproline, Ki(intercept) |
721590 |
6.3.3.6 | 1.1 |
- |
(3S,5S)-carbapenam 3-carboxylate |
pH 7.8, 22°C, variable substrate: (2S,5R)-carboxymethylproline, Ki(intercept) |
721590 |
6.3.3.6 | 1.3 |
- |
(3S,5S)-carbapenam 3-carboxylate |
pH 7.8, 22°C, variable substrate: (2S,5R)-carboxymethylproline, Ki(slope) |
721590 |
6.3.3.6 | 1.3 |
- |
(3S,5S)-carbapenam 3-carboxylate |
pH 7.8, 22°C, variable substrate: ATP, Ki(slope) |
721590 |
6.3.3.6 | 90 |
- |
L-proline |
pH 7.8, 22°C, variable substrate: (2S,5R)-carboxymethylproline, Ki(slope) |
721590 |
6.3.3.6 | 207 |
- |
L-proline |
pH 7.8, 22°C, variable substrate: ATP, Ki(intercept) |
721590 |