EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
    6.3.2.17 | 0.0000017 |
- |
Nalpha-(4-amino-4-deoxy-5,chloropteroyl)-L-ornithine |
- |
653856 |
| 6.3.2.17 | 0.0000031 |
- |
methotrexate-phosphinate |
Kis value, with methrotrexate as variable substrate, for recombinant enzyme |
649799 |
| 6.3.2.17 | 0.0000083 |
- |
Nalpha-(5,8-dideaza-5-chloropteroyl)-L-ornithine |
- |
653856 |
| 6.3.2.17 | 0.000018 |
- |
Nalpha-(4-amino-4-deoxy-8-deazapteroyl)-L-ornithine |
- |
653856 |
| 6.3.2.17 | 0.000056 |
- |
methotrexate-phosphinate |
Kii value, with methotrexate as variable substrate, for recombinant enzyme |
649799 |
| 6.3.2.17 | 0.000072 |
- |
Nalpha-(4-amino-4-deoxy-5,8-diazapteroyl)-L-ornithine |
- |
653856 |
| 6.3.2.17 | 0.000091 |
- |
2-[[[(3S)-3-[(4-[[(2-amino-4-oxo-3,4-dihydropteridin-6-yl)methyl]amino]benzoyl)amino]-3-carboxypropyl](hydroxy)phosphoryl]methyl]pentanedioic acid |
- |
705610 |
| 6.3.2.17 | 0.00015 |
- |
4-amino-4-deoxypteroyl-L-ornithine |
- |
653856 |
| 6.3.2.17 | 0.00035 |
- |
Nalpha-(5,8-dideazapteroyl)-L-ornithine |
- |
653856 |
| 6.3.2.17 | 0.00063 |
- |
2-[[(4-[[(2-amino-4-oxo-3,4-dihydropteridin-6-yl)methyl]amino]phenyl)(hydroxy)phosphoryl]methyl]pentanedioic acid |
- |
705610 |
