EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
5.4.99.7 | -999 |
- |
7-(4-allylmethylamino-but-2-ynyloxy)chromen-2-one |
above 0.1 mM |
662756 |
5.4.99.7 | -999 |
- |
7-(piperidinyl-N-hexyloxy)chromen-2-one |
above 0.1 mM |
662756 |
5.4.99.7 | 0.000013 |
- |
27-norsqualene |
pH 7.4, 37°C, liver microsomes |
727324 |
5.4.99.7 | 0.000015 |
- |
29-norsqualene |
pH 7.4, 37°C, liver microsomes |
727324 |
5.4.99.7 | 0.00002 |
- |
28-noroxidosqualene |
pH 7.4, 37°C, liver microsomes |
727324 |
5.4.99.7 | 0.00015 |
- |
7-[6-(allylmethylamino)-hexyloxy]-chromen-2-one |
- |
662756 |
5.4.99.7 | 0.00018 |
- |
7-[10-(allylmethylamino)-decyloxy]chromen-2-one |
- |
662756 |
5.4.99.7 | 0.00052 |
- |
7-[4'-(N-pyrrolidyn)-but-2-ynyloxy]chromen-2-one |
- |
662756 |
5.4.99.7 | 0.00104 |
- |
7-[6-(allylmethylamino)-hexyloxy]-chromen-2-one |
- |
662756 |
5.4.99.7 | 0.00104 |
- |
7-[8'(dimethylamino-N-octyloxy)]chromen-2-one |
- |
662756 |