EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
4.1.1.33 | 0.000049 |
- |
(R)-6-fluoromevalonate diphosphate |
wild type enzyme, at 30°C in 100 mM HEPES-NaOH (pH 7.0) |
715621 |
4.1.1.33 | 0.00005 |
- |
diphosphoglycolyl-L-proline |
pH and temperature not specified in the publication |
726990 |
4.1.1.33 | 0.000062 |
- |
6-fluoromevalonate 5-diphosphate |
wild type enzyme |
690629 |
4.1.1.33 | 0.00023 |
- |
6-fluoromevalonate diphosphate |
pH 7.0, 30°C |
748435 |
4.1.1.33 | 0.00058 |
- |
eriochrome black A |
wild-type, substrate (R)-5-diphosphomevalonate, pH 7.0, 30°C |
746911 |
4.1.1.33 | 0.00059 |
- |
Eriochrome Black T |
wild-type, substrate ATP, pH 7.0, 30°C |
746911 |
4.1.1.33 | 0.0012 |
- |
Eriochrome Black T |
wild-type, substrate (R)-5-diphosphomevalonate, pH 7.0, 30°C |
746911 |
4.1.1.33 | 0.0018 |
- |
eriochrome black A |
wild-type, substrate ATP, pH 7.0, 30°C |
746911 |
4.1.1.33 | 0.0023 |
- |
diphosphoglycolyl proline |
wild type enzyme |
690629 |
4.1.1.33 | 0.0027 |
- |
Eriochrome blue black |
wild-type, substrate (R)-5-diphosphomevalonate, pH 7.0, 30°C |
746911 |