EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.7.1.3 | 0.000005 |
- |
3-hydroxydeaminokynurenine |
- |
658345 |
3.7.1.3 | 0.000027 |
- |
(S)-(2-aminophenyl)-L-cysteine S,S-dioxide |
- |
660045 |
3.7.1.3 | 0.00003 |
- |
S-(2-aminophenyl)-L-cysteine dioxide |
wild-type enzyme, pH 8.0, 37ยฐC |
733832 |
3.7.1.3 | 0.00004 |
- |
3-hydroxydeaminokynurenine |
- |
658345 |
3.7.1.3 | 0.000055 |
- |
(4R)-5-bromodihydro-L-kynurenine |
- |
660045 |
3.7.1.3 | 0.0001 |
- |
3,7-dihydroxy-deamino-DL-kynurenine |
pH 7.9, at 37ยบC |
658605 |
3.7.1.3 | 0.0001 |
- |
3-hydroxydeaminokynurenine |
- |
658345 |
3.7.1.3 | 0.00017 |
- |
(4S)-5-bromodihydro-L-kynurenine |
- |
660045 |
3.7.1.3 | 0.00025 |
- |
3,5-dihydroxydeaminokynurenine |
- |
658345 |
3.7.1.3 | 0.0003 |
- |
(S)-(2-amino-4-bromophenyl)-L-cysteine S,S-dioxide |
- |
660045 |