EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.6.1.55 | 0.0000028 |
- |
6-(2,3-dichlorophenyl)-N4-methylpyrimidine-2,4-diamine |
at pH 7.5 and 37°C |
756449 |
3.6.1.55 | 0.000049 |
- |
8-oxo-dGMP |
pH 7.5, 23°C, Mg2+-activated, Ki(slope) |
654634 |
3.6.1.55 | 0.0000617 |
- |
8-bromo-7-deaza-dGTP |
at pH 7.5 and 37°C |
756449 |
3.6.1.55 | 0.000117 |
- |
8-chloro-7-deaza-dGTP |
at pH 7.5 and 37°C |
756449 |
3.6.1.55 | 0.000173 |
- |
8-oxo-dGMP |
pH 7.5, 23°C, Mn2+-activated, Ki(slope) |
654634 |
3.6.1.55 | 0.000203 |
- |
(S)-crizotinib |
at pH 7.5 and 37°C |
756449 |
3.6.1.55 | 0.000213 |
- |
7-deaza-dGTP |
at pH 7.5 and 37°C |
756449 |
3.6.1.55 | 0.000593 |
- |
8-oxo-dGMP |
pH 7.5, 23°C, Mn2+-activated, Ki(intercept) |
654634 |
3.6.1.55 | 0.00065 |
- |
7-iodo-7-deaza-dGTP |
at pH 7.5 and 37°C |
756449 |
3.6.1.55 | 0.00162 |
- |
8-oxo-dGMP |
pH 7.5, 23°C, Mg2+-activated, Ki(intercept) |
654634 |