EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.5.4.5 | 0.000025 |
- |
diazepinone riboside |
- |
669792 |
3.5.4.5 | 0.00006 |
- |
5-fluorozebularine |
tetramer of recombinant subunit CDA1, 37°C |
670747 |
3.5.4.5 | 0.0003 |
- |
5-fluorozebularine |
pH 7.5, 37°C, recombinant wild-type enzyme |
689935 |
3.5.4.5 | 0.0003 |
- |
5-fluorozebularine |
tetramer of recombinant subunit CDA2, 37°C |
670747 |
3.5.4.5 | 0.00042 |
- |
3,4,5,6-Tetrahydrouridine |
pH 7.5, 37°C, recombinant mutant R68Q |
689935 |
3.5.4.5 | 0.0006 |
- |
5-fluorozebularine |
pH 7.5, 37°C, recombinant mutant R68Q |
689935 |
3.5.4.5 | 0.00095 |
- |
zebularine |
pH 7.4, 37°C |
685915 |
3.5.4.5 | 0.0017 |
- |
5-fluorozebularine |
pH 7.5, 37°C, recombinant mutant Y60G |
689935 |
3.5.4.5 | 0.0067 |
- |
3,4,5,6-Tetrahydrouridine |
pH 7.5, 37°C, recombinant wild-type enzyme |
689935 |
3.5.4.5 | 0.007 |
- |
3,4,5,6-Tetrahydrouridine |
tetramer of recombinant subunit CDA1, 37°C |
670747 |