EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.24.34 | 0.0000007 |
- |
(2S,3R)-2-methyl-3-(2-methylpropyl)-1-(N-hydroxy)-4-(O-methyl)-L-tyrosine-N-methylamide |
pH 7.5, 37°C, BB-16 |
651879 |
3.4.24.34 | 0.000002 |
- |
(N-1(R)-carboxyethyl)-alpha-(S)-(4-phenyl-3-butynyl)glycyl-L-O-methyltyrosine, N-methylamide |
pH 7.5, 37°C, SA751 |
651879 |
3.4.24.34 | 0.00024 |
- |
(2R,S)-HONH-Mal(Me/Bn)-NH-CH2CH2CH2-Ph |
pH 7.6, 25°C |
652712 |
3.4.24.34 | 0.00038 |
- |
(2R,S)-HONH-Mal(Me/Bn)-NH-CH2CH2CH2CH2-Ph |
pH 7.6, 25°C |
652712 |
3.4.24.34 | 0.0011 |
- |
(2R,S)-HONH-Mal(Me/Bn)-NHBn |
pH 7.6, 25°C |
652712 |
3.4.24.34 | 0.0019 |
- |
(2R,S)-HONH-Mal(OH/Bn)-NHBn |
pH 7.6, 25°C |
652712 |
3.4.24.34 | 0.0023 |
- |
(2R,S)-HONH-Mal(NHAc/Bn)-NHBn |
pH 7.6, 25°C |
652712 |
3.4.24.34 | 0.0081 |
- |
(2R,S)-HONH-Mal(Me/Bn)-1,2,9,10-tetrahydroisoquinolide |
pH 7.6, 25°C |
652712 |
3.4.24.34 | 0.0096 |
- |
(2R,S)-HONH-Mal(Me/Bn)-NH-CH2CH2-Ph |
pH 7.6, 25°C |
652712 |
3.4.24.34 | 0.011 |
- |
(2R,S)-HONH-Mal(Me/Bn)-Oet |
pH 7.6, 25°C |
652712 |