EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
   3.4.23.39 | -999 |
- |
more |
Ki value for Iva-Val-Val-Sta-Ala-Sta is below 0.1 nM |
648188 |
| 3.4.23.39 | -999 |
- |
more |
Ki-values for (2S,5S,6R)-3-aza-5-hydroxy-7-phenyl-6-[(picolyl-L-valinyl)amino]-2-(m-(trifluoromethanesulfonylyxy)benzyl)-heptanoyl amide is above 2000 nM |
648186 |
| 3.4.23.39 | -999 |
- |
more |
the Ki-value for Ro17-7109 is above 0.015 mM |
648190 |
| 3.4.23.39 | 0.000000024 |
- |
pepstatin A |
- |
670126 |
| 3.4.23.39 | 0.000000037 |
- |
pepstatin |
pH 5.0, 37°C |
648187 |
| 3.4.23.39 | 0.00000004 |
- |
(5S,8S,12S,13S,16S,19S)-13-benzyl-12-hydroxy-8,23,23-trimethyl-16,19-bis(1-methylethyl)-5-(2-methylpropyl)-4,7,10,15,18,21-hexaoxo-3,6,9,14,17,20-hexaazatetracosan-1-amide |
- |
670126 |
| 3.4.23.39 | 0.00000007 |
- |
pepstatin A |
at pH 5.0 and 25°C |
753556 |
| 3.4.23.39 | 0.0000002 |
- |
N-[(3S)-3-[(2S,5S,14S)-14-[(3,3-dimethylbutanoyl)amino]-2-(1-methylethyl)-3,11,15-trioxo-1,4,10-triazacyclopentadecan-5-yl]-3-hydroxypropanoyl]-L-valyl-L-leucylglycinamide |
- |
670126 |
| 3.4.23.39 | 0.00000025 |
- |
benzyl [(1S,4S,5R,6R,7S,10S)-4,7-bis[(4-cyanophenoxy)methyl]-5,6-dihydroxy-1,10-bis(1-methylethyl)-2,9,12-trioxo-14-phenyl-13-oxa-3,8,11-triazatetradec-1-yl]carbamate |
- |
670126 |
| 3.4.23.39 | 0.0000005 |
- |
(4R)-3-[(2S,3S)-3-[[(2,6-dimethylphenoxy)acetyl]amino]-2-hydroxy-4-phenylbutanoyl]-N-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-5,5-dimethyl-1,3-thiazolidine-4-carboxamide |
- |
670126 |
