EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.23.34 | 0.0000002 |
- |
pepstatin A |
25°C, pH 4.0 |
670765 |
3.4.23.34 | 0.000003 |
- |
NYKDSCIG |
non-competitive |
699574 |
3.4.23.34 | 0.0000031 |
- |
pepstatin A |
40°C, pH 4.0, wild-type cathepsin E |
669151 |
3.4.23.34 | 0.000005 |
- |
SCGGIIIISCIA |
non-competitive |
699574 |
3.4.23.34 | 0.0000056 |
- |
pepstatin A |
40°C, pH 4.0, erythrocyte cathepsin E, hydrolysis of (7-methoxycoumarin-4-yl)acetyl-Gly-Ser-Pro-Ala-Phe-Leu-Ala-Lys(Dnp)-D-Arg-NH2 |
667861 |
3.4.23.34 | 0.00000582 |
- |
pepstatin A |
pH 3.5, 40°C, wild-type |
651797 |
3.4.23.34 | 0.00000606 |
- |
pepstatin A |
pH 3.5, 40°C, mutant D98E |
651797 |
3.4.23.34 | 0.00000648 |
- |
pepstatin A |
pH 3.5, 40°C, mutant T284S |
651797 |
3.4.23.34 | 0.0000078 |
- |
pepstatin A |
40°C, pH 4.0, gastric cathepsin E, hydrolysis of (7-methoxycoumarin-4-yl)acetyl-Gly-Ser-Pro-Ala-Phe-Leu-Ala-Lys(Dnp)-D-Arg-NH2 |
667861 |
3.4.23.34 | 0.0000084 |
- |
pepstatin A |
40°C, pH 4.0, erythrocyte cathepsin E, hydrolysis of (7-methoxycoumarin-4-yl)acetyl-Gly-Ser-Pro-Ala-Phe-Leu-Ala-Lys(Dnp)-D-Arg-NH2 |
667861 |