EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.22.36 | -999 |
- |
more |
the Ki-value for acetyl-IETD-aldehyde is below 6 nM and the Ki-value for acetyl-AEVD-aldehyde is below 12 nM |
647423 |
3.4.22.36 | 0.00000001 |
- |
cowpox serpin CrmA |
pH 7.5, 25°C |
647423 |
3.4.22.36 | 0.000000056 |
- |
acetyl-WEHD-aldehyde |
pH 7.5, 25°C |
647423 |
3.4.22.36 | 0.0000004 |
- |
NCGC00183434 |
in 50 mM HEPES, pH 7.4, containing 1 M sodium citrate, 100 mM NaCl, 0.1 mM EDTA, 10 mM dithiothreitol, 0.01% (v/v) CHAPS, 1% (v/v) DMSO, and 0.1 mg/ml bovine serum albumin |
708128 |
3.4.22.36 | 0.00000076 |
- |
acetyl-YVAD-aldehyde |
pH 7.5, 25°C |
647423 |
3.4.22.36 | 0.000001 |
- |
acetyl-YVAD-aldehyde |
pH 7.5, 37°C |
647724 |
3.4.22.36 | 0.000004 |
- |
(3S)-3-([6-(([3-methyl-4-(quinoxalin-2-ylamino)phenyl]carbonyl)amino)-2-thiophen-2-ylhexanoyl]amino)-4-oxobutanoic acid |
- |
667986 |
3.4.22.36 | 0.000004 |
- |
N-([4-(quinoxalin-2-ylamino)phenyl]carbonyl)-L-valyl-N-[(1S)-2-carboxy-1-formylethyl]-L-alaninamide |
- |
667986 |
3.4.22.36 | 0.000004 |
- |
N-acetyl-L-tyrosyl-alpha-glutamyl-N-[1-(carboxymethyl)-3-([dihydroxy(2-phenylethyl)-lambda4-sulfanyl]amino)-2-oxopropyl]-L-alaninamide |
- |
667948 |
3.4.22.36 | 0.000004 |
- |
N-[(benzyloxy)carbonyl]valyl-N-[1-(carboxymethyl)-3-([dihydroxy(2-phenylethyl)-lambda4-sulfanyl]amino)-2-oxopropyl]-L-alaninamide |
- |
667948 |