EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.21.76 | 0.00000012 |
- |
elafin |
25°C, recombinant elafin expressed in Pichia pastoris |
664822 |
3.4.21.76 | 0.00000012 |
- |
elafin |
methoxysuccinyl-lysyl-(2-picolinoyl)-Ala-Pro-Val-thiobenzylester as substrate, pH 7.4, 150 mM NaCl, 3 mM 4,4-dithiodipyridine |
664898 |
3.4.21.76 | 0.00000018 |
- |
trappin |
methoxysuccinyl-lysyl-(2-picolinoyl)-Ala-Pro-Val-thiobenzylester as substrate, pH 7.4, 150 mM NaCl, 3 mM 4,4-dithiodipyridine |
664898 |
3.4.21.76 | 0.00000018 |
- |
trappin-2 |
25°C, recombinant trappin-2 expressed in Pichia pastoris |
664822 |
3.4.21.76 | 0.000012 |
- |
serpin LEX032 |
pH 7.5, 25°C |
649534 |
3.4.21.76 | 0.000025 |
- |
elafin, oxidized with myeloperoxidase |
methoxysuccinyl-lysyl-(2-picolinoyl)-Ala-Pro-Val-thiobenzylester as substrate, pH 7.4, 150 mM NaCl, 3 mM 4,4-dithiodipyridine |
664898 |
3.4.21.76 | 0.000029 |
- |
elafin, oxidized with N-chlorosuccinimide |
methoxysuccinyl-lysyl-(2-picolinoyl)-Ala-Pro-Val-thiobenzylester as substrate, pH 7.4, 150 mM NaCl, 3 mM 4,4-dithiodipyridine |
664898 |
3.4.21.76 | 0.000035 |
- |
trappin, oxidized with myeloperoxidase |
methoxysuccinyl-lysyl-(2-picolinoyl)-Ala-Pro-Val-thiobenzylester as substrate, pH 7.4, 150 mM NaCl, 3 mM 4,4-dithiodipyridine |
664898 |
3.4.21.76 | 0.00005 |
- |
trappin, oxidized with N-chlorosuccinimide |
methoxysuccinyl-lysyl-(2-picolinoyl)-Ala-Pro-Val-thiobenzylester as substrate, pH 7.4, 150 mM NaCl, 3 mM 4,4-dithiodipyridine |
664898 |