EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.19.12 | -999 |
- |
more |
inhibition kinetics |
646099 |
3.4.19.12 | -999 |
- |
more |
inhibition kinetics of isatin O-acyl oximes, overview |
664573 |
3.4.19.12 | 0.0000001 |
- |
ubiquitin-aldehyde |
at 0.0006 mM ubiquitin, pH 7.8, 25°C |
646099 |
3.4.19.12 | 0.000001 |
- |
Ubiquitin aldehyde |
below, pH 7.5, 25°C, inhibition kinectis |
664127 |
3.4.19.12 | 0.0000023 |
- |
ubiquitin-aldehyde |
in absence of ubiquitin, pH 7.8, 25°C |
646099 |
3.4.19.12 | 0.00014 |
- |
ubiquitin |
- |
664127 |
3.4.19.12 | 0.00019 |
- |
ubiquitin |
- |
677540 |
3.4.19.12 | 0.0006 |
- |
ubiquitin |
pH 8.0, 37°C, isozyme L3 |
646091 |
3.4.19.12 | 0.00074 |
- |
3-amino-2-[(naphthalen-2-yloxy)carbonyl]-6-oxo-6,7-dihydrothieno[2,3-b]pyridine-5-carboxylic acid |
- |
678672 |
3.4.19.12 | 0.00091 |
- |
3-amino-2-[(4-methylphenyl)carbonyl]-6-oxo-6,7-dihydrothieno[2,3-b]pyridine-5-carboxylic acid |
- |
678672 |