EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.17.21 | 0.000000003 |
- |
(S)-2-(3-((S)-1-carboxy-(4-iodobenzamido)pentyl)ureido)pentanedioic acid |
pH and temperature not specified in the publication |
754372 |
3.4.17.21 | 0.0000000086 |
- |
(S)-2-(3-((S)-5-(N-(4-bromobenzyl)-6-(4-(4-(4-(4-carboxy-3-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoyl)piperazin-1-yl)phenyl)-piperazin-1-yl)nicotinamido)-1-carboxypentyl)ureido)pentanedioic acid |
pH and temperature not specified in the publication |
754372 |
3.4.17.21 | 0.00000001 |
- |
N-([(1S)-1-carboxy-5-([(4-iodophenyl)carbonyl]amino)pentyl]carbamoyl)-L-glutamic acid |
pH not specified in the publication, temperature not specified in the publication |
731449 |
3.4.17.21 | 0.000000017 |
- |
N-[[(1S)-1-carboxy-5-(4-iodobenzamido)pentyl]carbamoyl]-L-glutamic acid |
37°C, pH 7.4 |
753584 |
3.4.17.21 | 0.000000018 |
- |
DKFZ-PSMA-11 |
pH and temperature not specified in the publication |
754372 |
3.4.17.21 | 0.000000018 |
- |
N-[[(1S)-1-carboxy-5-([5-[3-(3-[[[2-[[[5-(2-carboxyethyl)-2-hydroxyphenyl]methyl](carboxymethyl)amino]ethyl](carboxymethyl)amino]methyl]-4-hydroxyphenyl)propanamido]pentanoyl]amino)pentyl]carbamoyl]-L-glutamic acid |
37°C, pH 7.4 |
753584 |
3.4.17.21 | 0.000000021 |
- |
N-[[(1S)-5-([(4-bromophenyl)methyl][6-[4-(4-[4-[4-carboxy-3-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoyl]piperazin-1-yl]phenyl)piperazin-1-yl]pyridine-3-carbony]amino)-1-carboxypentyl]carbamoyl]-L-glutamic acid |
37°C, pH 7.4 |
753584 |
3.4.17.21 | 0.000000028 |
- |
N-[[(1S)-1-carboxy-5-(4-iodobenzamido)pentyl]carbamoyl]-L-glutamic acid |
37°C, pH 7.4 |
753584 |
3.4.17.21 | 0.000000049 |
- |
(S)-2-(3-((S)-5-(6-(4-(4-(4-acetylpiperazin-1-yl)phenyl)piperazin-1-yl)-N-(4-bromobenzyl)nicotinamido)-1-carboxypentyl)ureido)-pentanedioic acid |
pH and temperature not specified in the publication |
754372 |
3.4.17.21 | 0.000000049 |
- |
N-[[(1S)-5-([(4-bromophenyl)methyl][6-[4-(4-[4-[4-carboxy-3-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoyl]piperazin-1-yl]phenyl)piperazin-1-yl]pyridine-3-carbony]amino)-1-carboxypentyl]carbamoyl]-L-glutamic acid |
37°C, pH 7.4 |
753584 |